amprenavir


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Related to amprenavir: Fosamprenavir, Atazanavir
Translations

amprenavir

n amprenavir m
References in periodicals archive ?
Previously, within the biopharmaceutical industry, Dr McGowan was a senior research physician at GlaxoSmithKline in the UK where he contributed to the development of the antiviral drugs Amprenavir and Abacavir.
(31) Additionally, amprenavir, LPV/r, and ritonavir demonstrated more glucose uptake inhibition via blockade of the glucose transporter type 4 than ATV.
(48) Other PIs such as nelfinavir, amprenavir, saquinavir, ritonavir, and darunavir have also been reported to cause urolithiasis.
The first generation of HIV protease inhibitors, including Saquinavir (1), Ritonavir (2) Nelfinavir (3), Indinavir (4), and Amprenavir (5) (Figure 4), was initially effective against HIV infection; the fast-emerging resistance to these agents has been a substantial and persistent problem in the treatment of AIDS.
More recently, they are used in treatment of Alzheimer's disease [14], Amprenavir belongs to this class and is utilized as anti-HIV protease inhibitor [15] and also as anti-cancer agent [16].
(20) This University of Sao Paulo group gives the second-generation PIs--ritonavir-boosted lopinavir, amprenavir, fosamprenavir, and tipranavir--the worst dyslipidemia marks in their Table 2 summary: three up-arrows indicating the greatest likelihood of spawning dyslipidemia.
In a glioblastoma cell line, HIV Protease Inhibitors--Nelfinavir and Amprenavir reduced the expression of vascular endothelial growth factor (VEGF) and hypoxia inducible factor-alpha (Pore et al., 2006).
The other prescribed PIs were RTV-boosted lopinavir (LPV) (3.0%), RTV-boosted amprenavir (APV) (2.0%), atazanavir (ATV) (1.0%), and saquinavir (SQV) (1.0%).
[19] Nevirapine, delavirdine and efavirenz, abacavir, amprenavir cause rashes frequently due to hypersensitivity which usually resolve spontaneously.
Possible linkage of amprenavir with intracranial bleeding in an HIV-infected hemophiliac.
Moderate CYP3A4 inhibitors include amprenavir, atazanavir, ciprofloxacin, diltiazem, erythromycin, fluconazole, fosamprenavir, verapamil, and grapefruit juice.
Se evaluaron un total de 13418 compuestos obtenidos de la libreria PubChem con estructuras similares a A70 (1407), Pepstatin A (7280), Amprenavir (589), Indinavir (1519), Ritonavir (1623) y Saquinavir (1000).